Posaconazole 171228-49-2 Antibiyotike
Kwishura:T / T, L / C.
Inkomoko y'ibicuruzwa:Ubushinwa
Icyambu cyo kohereza:Beijing / Shanghai / Hangzhou
Ubushobozi bwo gukora:20kg / ukwezi
Tegeka (MOQ):10g
Igihe cyo kuyobora:Iminsi y'akazi
Imiterere y'ububiko:Ubitswe ahantu hakonje, humye, ubushyuhe bwicyumba.
Ibikoresho bipakira:vial
Ingano yububiko:10g / vial
Amakuru yumutekano:Ntabwo ari ibintu biteje akaga
Intangiriro
Posaconazole numuti wa triazole antifungal.
Posaconazole ikoreshwa mu kuvura indwara ziterwa na Aspergillus na Candida.Irakoreshwa kandi mukuvura kandidiasis ya oropharyngeal (OPC), harimo na OPC yanga itraconzaole na / cyangwa kuvura fluconazole.
Ikoreshwa kandi mu kuvura indwara zandurira mu bwoko bwa Candida, Mucor, na Aspergillus ku barwayi badafite ubudahangarwa bukabije.
Ibisobanuro (munzu isanzwe)
Ingingo | Ibisobanuro |
Kugaragara | Ifu yera cyangwa hafi yera, ifu ya hygroscopique |
Ingingo | Ibisobanuro |
Kugaragara | Ifu yera cyangwa yera-ifu ya kristaline |
Kuzenguruka byihariye | -28.0 ° ~ -34.0 ° |
Ifishi ya kirisiti | Igomba kuba kristaline Ⅰ, hamwe na 2-ya nguni ya 14.4 ± 0.2 °, 19.2 ± 0.2 °, 21.7 ± 0.2 °, 24.3 ± 0.2 ° 29.3 ± 0.2 ° |
Kumenyekanisha | IR, HPLC |
Ibintu bifitanye isano I. | PO-R1 NMT 0,10% |
PO-R2 NMT 0,10% | |
PO-R3 NMT 0,10% | |
PO-R4 NMT 0,10% | |
PO-D3 & PO-D5 NMT 0,10% | |
PO-D7 & PO-D10 NMT 0,10% | |
Buriwese wanduye NMT 0,10% | |
Umwanda wose NMT 0.5% | |
Ibintu bifitanye isano Ⅱ | PO-E NMT 0,10% |
PO-D1 NMT 0,10% | |
PO-R5 NMT 0,10% | |
Amashanyarazi asigaye | Methanol NMT 3000ppm |
Ethanol NMT 5000ppm | |
Dichloromethane NMT 600ppm | |
Tetrahydrofuran NMT 720ppm | |
N, N-dimethyl formamide NMT 880ppm | |
Triethylamine NMT 100ppm | |
Dimethy sulfoxide NMT 5000ppm | |
Amazi | NMT 2.0% |
Ibisigisigi byo gutwikwa | NMT 0.1% |
Ibyuma biremereye | NMT 10ppm |
Imipaka ntarengwa | Indege yose NMT 1000cfu / g Imisemburo yose hamwe na NMT 100cfu / g E.coli igomba kuba idahari |
Suzuma | 98.0% -102.0% (ku buryo budasanzwe) |
98.0% -102.0% (kuri anhydrous na solvents kubuntu) |