Pimobendan 74150-27-9 Metabolism PDE inhibitor
Kwishura:T / T, L / C.
Inkomoko y'ibicuruzwa:Ubushinwa
Icyambu cyo kohereza:Beijing / Shanghai / Hangzhou
Tegeka (MOQ):1g
Igihe cyo kuyobora:Iminsi 3 y'akazi
Ubushobozi bwo gukora:1kg / ukwezi
Imiterere y'ububiko:Ubitswe ahantu hakonje, humye, ubushyuhe bwicyumba.
Ibikoresho bipakira:vial, icupa
Ingano yububiko:1g / vial, 5 / vial, 10g / vial, 50g / icupa, 500g / icupa
Amakuru yumutekano:UN 2811 6.1 / PG 3
Intangiriro
Pimobendan, ni imiti yamatungo.Ni sensibilisiyumu ya calcium kandi ihitamo inhibitori ya fosifisiyose 3 (PDE3) ifite ingaruka nziza za inotropique na vasodilator.
Pimobendan ikoreshwa mugucunga kunanirwa k'umutima ku mbwa, bikunze guterwa n'indwara ya myxomatous mitral valve (nanone izwi nka endocardiose), cyangwa umutima wagutse.Ubushakashatsi bwerekanye ko nka mitiweli, pimobendan yongera igihe cyo kubaho kandi igateza imbere ubuzima bw’abarwayi ba kineine bafite ikibazo cyo kunanirwa k'umutima cya kabiri kugeza ku ndwara ya mitral iyo ugereranije na benazepril, inhibitori ya ACE.
Ibisobanuro (USP43)
Ingingo | Ibisobanuro |
Kugaragara | Ifu yera cyangwa yumuhondo gato, hygroscopique |
Mp | Hafi ya 242 ℃ |
Gukemura | Mubyukuri bidashobora gushonga mumazi, gushonga kubusa muri dimethylformamide, gushonga gake muri acetone na methanil. |
Kumenyekanisha | Infrared absorption spectrophotometrie, Kugereranya pimobendan CRS. |
Igihe cyo kugumana impinga nyamukuru yikibazo cyicyitegererezo gihuye nicyo gisubizo cyibisanzwe, nkuko byabonetse mubizamini bya Organic Impurities. | |
Ibyuma biremereye | ≤10ppm |
Ubunini | P90 ≤ 25μ m |
Ingano ya Particle | 20-80 mesh |
Amashanyarazi asigaye | ≤ 500ppm |
Amazi | ≤ 1.0% |
Suzuma | 98.0% ~ 102.0% |
Ivu | ≤ 0,10% |
Ibintu bifitanye isano (HPLC) | |
umwanda A. | ≤ 0,10% |
umwanda B. | ≤ 0,10% |
Ibindi byose byanduye | ≤ 0,10% |
Umwanda wuzuye | ≤ 0,20% |