Imiyoboro ya Laboratoire

Ibicuruzwa

Mirabegron 223673-61-8 Inhibitor Ikimenyetso cya Neuronal

Ibisobanuro bigufi:

Synonyme:YM 178, N- (4- (2-

CAS No.:223673-61-8

Ubwiza:mu nzu

Inzira ya molekulari:C21H24N4O2S

Uburemere bwa formula:396.51


Ibicuruzwa birambuye

Ibicuruzwa

Kwishura:T / T, L / C.
Inkomoko y'ibicuruzwa:Ubushinwa
Icyambu cyo kohereza:Beijing / Shanghai / Hangzhou
Ubushobozi bwo gukora:100kg / ukwezi
Tegeka (MOQ):25kg
Igihe cyo kuyobora:Iminsi y'akazi
Imiterere y'ububiko:Ubitswe ahantu hakonje, humye, ubushyuhe bwicyumba.
Ibikoresho bipakira:ingoma
Ingano yububiko:25kg / ingoma
Amakuru yumutekano:Ntabwo ari ibintu biteje akaga

Mirabegron

Intangiriro

Mirabegron, ni beta-3 adrenergic reseptor agonist, itera beta-3 adrenergic reseptor kandi ikoroshya imitsi yoroshye ya detrusor, bityo ikongerera ubushobozi bwuruhago kandi ikoreshwa mukuvura ibimenyetso byuruhago rukabije (OAB), nko gusaba kwifata, byihutirwa, n'inshuro.

Ibyiza byayo bisa n'imiti igabanya ubukana nka solifenacin cyangwa tolterodine.

Ibisobanuro (USP / EP)

Ingingo

Ibisobanuro

Kugaragara Umweru kugeza ifu yera

Kumenyekanisha

IR, HPLC
Ibirimo amazi NMT 0.5%
Ibisigisigi byo gutwikwa NMT 0.1%
Icyuma kiremereye NMT 20ppm
Ibirimo Palladium NMT 20ppm
Isomer NTM 0.5%
Ibintu bifitanye isano Z-168 *: NMT 0.15%
  SC03610 *: NMT 0.15%
  Ibindi byose bitanduye: NMT 0,10%
  Umwanda wose: NMT 0.5%
2- (2-aminothianzol-4-yl) aside aside NMT 0.1%
Ibisigisigi Methanol: NMT 0.3%
  Ethyl acetate: NMT 0.5%
  THF: NMT 0.072%
  Benzene: NMT 0.0002%
  Toluene: NMT 0.089%
Suzuma 98.0% - 102.0%
PSD D (0.5): 10 mm - 30 mm
  D (0.9): 20 mm - 80 mm

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