Imiyoboro ya Laboratoire

Ibicuruzwa

Doramectin 117704-25-3 Antibiyotike Irwanya Parasitike

Ibisobanuro bigufi:

Synonyme:25-Cclohexyl-avermectin B1, Avermectin A1a

CAS No.:117704-25-3

Ubwiza:mu nzu

Inzira ya molekulari:C50H74O14

Uburemere bwa formula:899.11


Ibicuruzwa birambuye

Ibicuruzwa

Kwishura:T / T, L / C.
Inkomoko y'ibicuruzwa:Ubushinwa
Icyambu cyo kohereza:Beijing / Shanghai / Hangzhou
Ubushobozi bwo gukora:15kg / ukwezi
Tegeka (MOQ):1kg
Igihe cyo kuyobora:Iminsi y'akazi
Imiterere y'ububiko:Bika ku bushyuhe 2-8 ℃ igihe kirekire, urinzwe n'umucyo.
Ibikoresho bipakira:icupa
Ingano yububiko:1kg / ingoma
Amakuru yumutekano:UN 2811 6.1 / PG 3

Doramectin

Intangiriro

Dorametin ni igisekuru gishya imiti ya antiparasitike ya macrolide.Ni antibiyotike ya avermectin ikorwa na fermentation yubwoko bushya bwa Streptomyces avermitis hamwe na acide cyclohexamic nkibibanziriza.Bifatwa nkimwe mumiti myiza ya antiparasitike mumuryango wa avermectin.

Ingaruka zo kurwanya udukoko twa Doramectin zisa na Ivermectin, zishobora kubuza kwanduza imitsi imitsi hagati y'imitsi n'imitsi, kandi bigatuma udukoko twamugaye tugapfa kure yabakiriye.Nyamara, kubera umuvuduko mwinshi wamaraso ya doramectine mumubiri, kurandura biratinda cyane, kandi igihe cyo gufata neza igihe kirekire, bityo ingaruka zo kurwanya udukoko ni nziza kuruta Ivermectin.Kuberako nta reaction ya allergique iyo ukoresheje Doramectin, bityo rero ni umutekano kurushaho gukoreshwa.Bifatwa kandi nk'ibiyobyabwenge aho kuba Ivermectin.

Ikoreshwa mukuvura no kugenzura parasitose y'imbere (gastrointestinal na pulmonary nematode), amatiku na mange (hamwe na ectoparasite).

Mubuvuzi bwerekana ko Doramectin igira ingaruka nziza kuri nematode mu nzira yigifu yingurube.Nk’uko raporo ibigaragaza, ingurube zatanzwe mu buryo butemewe ku gipimo cya 0.3 mg / kg cy'umubiri.Ubwiyongere bwibiro byubwandu bwanduye nibisanzwe byanduye byari hejuru cyane ugereranije nitsinda rishinzwe kugenzura iminsi 7, 14 na 21 nyuma yubuyobozi.Ugereranije nitsinda rishinzwe kugenzura, inyo zavanyweho 100% nta ngaruka mbi.

Irerekana kandi mubuvuzi mukuvura ibisebe bya Sarcoptes, hari ingaruka nziza zonsa ingurube kugeza kubiba.

Doramectin iraboneka kandi kumafarasi nka gel yo munwa, uburyohe, bioadhesive gel mwizina.

Doramectin ntabwo ihindagurika muri kamere.Irabora vuba kandi idakora munsi yizuba.Imiti yacyo isigaye ni uburozi ku mafi n’ibinyabuzima byo mu mazi.Kubwibyo, hakwiye kwitabwaho kurinda amazi.

Ibisobanuro (Mu nzu isanzwe)

Ingingo

Ibisobanuro

Kugaragara Ifu ya kirisiti yera
Kumenyekanisha HPLC, IR
Kugaragara kw'igisubizo Igisubizo kirasobanutse kandi ntabwo gifite amabara menshi kuruta igisubizo BY6
Amazi ≤3%
Icyuma kiremereye ≤20ppm
Ashu ≤0.1%
BHT 0002000ppm
Ibintu bifitanye isano Avermectin B1a≤1.5%
Avermectin B1b≤1.0%
Avermectin B1a na Avermectin B1b≤2.0%
Umwanda wose NMT 5.0%
Ibisigisigi Acetone≤5000ppm
Ethanol≤30000ppm
Ethyl acetate≤5000ppm
Methanol≤3000ppm
Suzuma ≥95% (kuri anhydrous na solvent kubuntu)

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